Information about Crestor (Rosuvastatin)
Crestor is a medication that belongs to the statin class of drugs, used primarily to lower cholesterol levels in the blood. Rosuvastatin, the active ingredient, works by inhibiting HMG-CoA reductase, an enzyme involved in cholesterol synthesis in the liver. This action helps to reduce levels of low-density lipoprotein (LDL) cholesterol and triglycerides while increasing high-density lipoprotein (HDL) cholesterol.
Product Highlights
- Effective in reducing cardiovascular risk, it is used for managing hyperlipidemia and preventing heart attacks and strokes.
- Available in various strengths, Crestor offers flexible dosing options and is well-tolerated with a robust safety profile.
Key Ingredient
Key Benefits
- Significantly lowers LDL cholesterol and triglycerides, and raises HDL cholesterol.
- Helps in preventing heart attacks, strokes, and other cardiovascular events.
- Available in various strengths (5 mg, 10 mg, 20 mg, 40 mg), allowing tailored treatment based on individual needs.
Direction of Use
- Taken orally, with or without food.
- Typically starts at 10 mg once daily, with the dose adjusted based on individual response and treatment goals. The highest recommended daily dose is 40 mg.
Safety Concerns
- Potential for muscle pain, tenderness, or weakness; risk of rhabdomyolysis (a serious muscle condition) is higher at higher doses.
- May cause liver enzyme elevations; liver function should be monitored periodically.
- Can interact with other medications, including certain anticoagulants and other drugs metabolized by CYP3A4.
Avoid Crestor (Rosuvastatin) If
- Avoid if there is a known hypersensitivity to rosuvastatin or any other component of the medication.
- Use is contraindicated in patients with active liver disease or unexplained persistent elevations of liver enzymes.
- Not advised for use during pregnancy or breastfeeding due to potential risks to the fetus or infant.
